產品描述
A-674563 is an Akt1 inhibitor with Ki of 11 nM, modest potent to PKA and >30-fold selective for Akt1 over PKC
產品價格
貨號 | 規格 | 價格 |
CC2826 |
2mg |
1036.00 元 |
CC2826 | 5mg | 1952.00 元 |
CC2826 | 10mg | 3463.00 元 |
化學數據
分子量Molecular Weight (MW) | 358.44 | |
---|---|---|
化學式Formula |
C22H22N4O |
|
CAS號CAS No. | 552325-73-2 | |
溶解性Solubility (25°C) | 二甲基亞砜DMSO |
72 mg/mL(200.87 mM) |
水Water | 72 mg/mL(200.87 mM) | |
乙醇Alcohol | 18 mg/mL(50.21 mM) |
制備儲備液
濃度/溶劑體積(DMSO)/質量 | 1 mg | 5 mg | 10 mg |
1 mM | 2.7899 mL | 13.9493 mL | 27.8987 mL |
5 mM | 0.5580 mL | 2.7899 mL | 5.5797 mL |
10 mM | 0.2790 mL | 1.3949 mL | 2.7899 mL |
50 mM | 0.0558 mL | 0.2790 mL | 0.5580 mL |